Receptors in the training set

278 receptors, 333,727 fitting measurements and 19,393 held-out measurements. Generated from the measurement files the models were built from, so it cannot drift from the training set.

Gene symbols link to GeneCards and accessions to UniProt. The two accuracy columns are that receptor's own held-out accuracy, with the number of comparisons it rests on beside it. A receptor with a handful of comparisons can read 0.000 or 1.000 and neither means much, so read the count. A dash means the model was not scored on that receptor.

Every column heading sorts, except endpoints. Click once for descending, again for ascending. The default is fitting measurements, largest first.

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Minimum held-out comparisons

#▾	Gene▾	Accession▾	Fit measurements▾	Fit ligands▾	Held-out▾	Potency accuracy▾	Potency n▾	Selectivity accuracy▾	Selectivity n▾	Endpoints
1	DRD2	P14416	11,538	10,284	863	0.637	13,624	0.782	1,628	Ki 9483, IC50 1051, EC50 743, Kb 161, Kd 100
2	CNR2	P34972	10,595	9,317	621	0.650	11,493	0.887	266	Ki 4926, EC50 4237, IC50 1406, Kb 14, Kd 12
3	CNR1	P21554	9,624	8,598	554	0.696	9,189	0.848	309	Ki 4034, EC50 3665, IC50 1655, Kd 188, Kb 82
4	OPRM1	P35372	9,596	7,987	869	0.573	12,148	0.662	890	Ki 6305, EC50 1756, IC50 1454, Kb 47, Kd 34
5	HCRTR2	O43614	8,592	7,996	1,025	0.695	14,882	0.881	666	IC50 5109, Ki 2267, EC50 1027, Kd 146, Kb 43
6	ADORA2A	P29274	8,506	8,050	382	0.770	8,632	0.673	294	Ki 6490, IC50 1606, EC50 320, Kd 76, Kb 14
7	HCRTR1	O43613	7,577	7,221	708	0.761	9,981	0.881	665	IC50 4935, Ki 2189, EC50 271, Kd 151, Kb 31
8	OPRK1	P41145	7,540	6,374	492	0.602	12,399	0.635	761	Ki 4365, IC50 1571, EC50 1533, Kb 56, Kd 15
9	HTR1A	P08908	7,082	6,260	266	0.723	6,564	0.729	993	Ki 5476, EC50 789, IC50 696, Kd 68, Kb 53
10	HTR2A	P28223	6,806	6,218	632	0.693	11,235	0.695	1,536	Ki 4971, IC50 1217, EC50 577, Kb 37, Kd 4
11	DRD3	P35462	6,669	6,060	698	0.749	11,576	0.777	1,510	Ki 5824, EC50 481, IC50 301, Kb 37, Kd 26
12	OPRD1	P41143	6,619	5,586	385	0.692	8,912	0.732	381	Ki 4453, IC50 1127, EC50 979, Kb 43, Kd 17
13	ADORA1	P30542	6,545	6,135	156	0.716	4,748	0.710	262	Ki 5149, IC50 817, EC50 407, Kd 165, Kb 7
14	ADORA3	P0DMS8	6,332	5,809	258	0.538	7,414	0.648	199	Ki 5080, IC50 935, EC50 216, Kd 63, Kb 38
15	HRH3	Q9Y5N1	5,536	4,701	118	0.695	5,073	0.653	176	Ki 4008, IC50 800, EC50 378, Kd 273, Kb 77
16	HTR6	P50406	5,262	4,522	348	0.608	7,154	0.761	808	Ki 3920, IC50 897, Kb 246, EC50 122, Kd 77
17	ADORA2B	P29275	5,119	4,877	153	0.556	5,587	0.566	166	Ki 2759, IC50 1847, EC50 429, Kb 48, Kd 36
18	HTR2C	P28335	4,791	4,347	359	0.604	10,323	0.684	1,122	Ki 2811, EC50 999, IC50 972, Kb 7, Kd 2
19	MC4R	P32245	4,284	3,234	113	0.679	2,176	0.670	191	Ki 2027, EC50 1360, IC50 851, Kd 29, Kb 17
20	S1PR1	P21453	4,087	3,687	93	0.622	2,562	0.717	106	EC50 2658, IC50 1280, Ki 139, Kd 9, Kb 1
21	GRM5	P41594	3,958	3,461	100	0.568	2,817	0.556	9	IC50 2042, EC50 1325, Ki 579, Kb 10, Kd 2
22	MCHR1	Q99705	3,917	3,665	55	0.569	752	1.000	12	IC50 2177, Ki 1605, Kb 66, EC50 66, Kd 3
23	PTGDR2	Q9Y5Y4	3,801	3,544	4	0.000	2	1.000	3	IC50 2102, Ki 1433, EC50 254, Kb 7, Kd 5
24	APLNR	P35414	3,675	3,493	40	0.521	445	0.525	200	EC50 3310, Ki 264, IC50 100, Kd 1
25	CHRM1	P11229	3,651	3,470	92	0.663	1,381	0.574	413	Ki 1559, EC50 966, IC50 885, Kb 161, Kd 80
26	DRD4	P21917	3,581	3,179	181	0.699	5,668	0.726	752	Ki 2857, IC50 378, EC50 331, Kd 13, Kb 2
27	HTR7	P34969	3,564	3,351	186	0.722	4,959	0.762	1,000	Ki 2768, IC50 482, EC50 240, Kb 65, Kd 9
28	OPRL1	P41146	3,382	2,950	56	0.564	835	0.796	108	Ki 2219, IC50 718, EC50 375, Kb 58, Kd 12
29	CHRM3	P20309	3,164	3,011	154	0.713	4,963	0.571	387	Ki 1937, IC50 974, EC50 154, Kd 99
30	TACR1	P25103	2,899	2,767	2	—	—	0.929	14	IC50 1817, Ki 951, Kd 113, EC50 16, Kb 2
31	CHRM2	P08172	2,825	2,609	179	0.736	4,978	0.646	469	Ki 1667, IC50 589, EC50 225, Kb 191, Kd 153
32	FFAR1	O14842	2,679	2,506	184	0.672	4,892	0.500	2	EC50 2419, Ki 142, IC50 107, Kd 11
33	S1PR3	Q99500	2,641	2,598	5	0.500	2	1.000	7	EC50 1778, IC50 850, Kd 8, Ki 5
34	ADRB2	P07550	2,515	2,160	258	0.770	8,613	0.591	462	EC50 1053, IC50 677, Ki 639, Kd 143, Kb 3
35	CCR5	P51681	2,468	2,428	53	0.627	1,288	0.000	22	IC50 2237, Ki 157, EC50 60, Kd 14
36	GHSR	Q92847	2,438	1,969	20	0.528	72	1.000	1	IC50 960, EC50 730, Ki 667, Kb 78, Kd 3
37	CHRM4	P08173	2,295	2,200	162	0.662	5,617	0.650	363	Ki 1363, EC50 624, IC50 272, Kb 28, Kd 8
38	HTR2B	P41595	2,288	2,033	280	0.696	5,890	0.729	889	Ki 1551, EC50 471, IC50 242, Kb 23, Kd 1
39	CRHR1	P34998	2,271	2,132	0	—	—	—	—	Ki 1482, IC50 696, EC50 85, Kd 8
40	CCR2	P41597	2,263	2,178	24	0.628	231	0.043	23	IC50 1928, Ki 307, Kd 19, EC50 9
41	GRM2	Q14416	2,246	2,007	125	0.664	4,445	0.793	29	EC50 1046, IC50 944, Ki 197, Kd 45, Kb 14
42	HRH4	Q9H3N8	2,200	1,812	21	0.898	167	0.887	53	Ki 1556, EC50 307, IC50 167, Kd 145, Kb 25
43	HRH1	P35367	2,147	2,022	146	0.704	3,868	0.683	587	Ki 1553, IC50 339, Kd 158, Kb 51, EC50 46
44	FPR2	P25090	2,133	2,039	350	0.522	9,847	0.667	81	EC50 1408, Kd 370, IC50 326, Ki 29
45	ADRA1A	P35348	2,132	2,022	116	0.640	2,468	0.702	728	Ki 1513, EC50 293, IC50 292, Kd 21, Kb 13
46	DRD1	P21728	1,924	1,774	149	0.734	5,220	0.732	680	Ki 1443, EC50 288, IC50 148, Kd 35, Kb 10
47	ADRB1	P08588	1,901	1,780	112	0.706	2,062	0.730	270	EC50 806, IC50 611, Ki 411, Kd 72, Kb 1
48	AVPR1A	P37288	1,900	1,652	274	0.679	8,661	0.877	65	Ki 997, IC50 677, EC50 196, Kb 21, Kd 9
49	CXCR3	P49682	1,896	1,824	42	0.377	629	1.000	5	IC50 1567, Ki 291, EC50 35, Kd 3
50	CCKBR	P32239	1,868	1,720	5	—	—	—	—	IC50 1245, Ki 505, EC50 110, Kd 8
51	GRM4	Q14833	1,825	1,756	9	0.500	18	0.550	20	EC50 1637, IC50 96, Ki 78, Kb 14
52	GNRHR	P30968	1,792	1,680	5	1.000	4	1.000	1	IC50 1020, Ki 733, Kd 38, Kb 1
53	ADRA1B	P35368	1,790	1,722	76	0.644	1,796	0.679	638	Ki 1400, EC50 225, IC50 147, Kd 13, Kb 5
54	GPR119	Q8TDV5	1,749	1,683	82	0.645	2,024	0.524	185	EC50 1680, Ki 48, IC50 21
55	ADRB3	P13945	1,703	1,611	72	0.554	772	0.753	215	EC50 1300, Ki 318, IC50 58, Kd 27
56	EDNRA	P25101	1,702	1,633	53	0.528	1,177	1.000	11	IC50 1377, Ki 240, Kb 68, EC50 12, Kd 5
57	SSTR4	P31391	1,655	1,434	140	0.699	4,018	0.842	95	EC50 613, IC50 573, Ki 438, Kd 31
58	GLP1R	P43220	1,652	1,451	392	0.670	5,013	0.579	209	EC50 1343, IC50 244, Ki 56, Kd 9
59	MC1R	Q01726	1,634	1,145	97	0.655	1,671	0.615	174	EC50 788, Ki 524, IC50 318, Kd 4
60	HTR1D	P28221	1,629	1,459	54	0.507	1,378	0.680	519	Ki 1125, IC50 347, EC50 145, Kb 9, Kd 3
61	MC5R	P33032	1,626	1,367	38	0.670	173	0.847	98	IC50 846, Ki 436, EC50 340, Kd 4
62	SSTR2	P30874	1,577	1,538	87	0.780	1,070	0.648	91	Ki 564, IC50 501, EC50 476, Kd 36
63	MC3R	P41968	1,569	1,119	88	0.669	1,424	0.726	190	Ki 657, EC50 535, IC50 356, Kd 21
64	ACKR3	P25106	1,564	1,521	59	0.599	1,185	0.882	17	IC50 821, EC50 649, Ki 94
65	PTGER4	P35408	1,555	1,298	111	0.557	4,878	0.965	57	IC50 641, Ki 591, EC50 267, Kb 49, Kd 7
66	FFAR4	Q5NUL3	1,535	1,533	39	0.581	391	0.486	107	EC50 1533, IC50 2
67	ADRA1D	P25100	1,534	1,469	54	0.602	1,122	0.655	501	Ki 1156, EC50 214, IC50 159, Kb 5
68	TACR3	P29371	1,518	1,247	44	0.547	848	—	—	Ki 897, IC50 474, EC50 123, Kb 13, Kd 11
69	P2RY12	Q9H244	1,490	1,289	14	0.894	47	0.500	6	IC50 752, Ki 650, EC50 81, Kb 4, Kd 3
70	HTR1B	P28222	1,458	1,372	73	0.636	1,236	0.675	584	Ki 1060, IC50 303, EC50 79, Kb 8, Kd 8
71	NPY5R	Q15761	1,435	1,363	23	1.000	20	0.938	32	IC50 791, Ki 606, EC50 33, Kb 5
72	CHRM5	P08912	1,404	1,375	127	0.515	2,552	0.512	422	Ki 877, IC50 320, EC50 203, Kd 4
73	MTNR1A	P48039	1,400	1,184	66	0.676	1,412	0.873	63	Ki 962, IC50 232, EC50 179, Kb 25, Kd 2
74	GCGR	P47871	1,379	1,315	34	0.597	489	0.795	39	IC50 868, Ki 304, EC50 151, Kb 56
75	CXCR4	P61073	1,324	1,196	154	0.457	4,696	0.778	9	IC50 1103, EC50 200, Ki 16, Kb 4, Kd 1
76	F2RL3	Q96RI0	1,320	1,207	40	0.661	768	0.950	20	IC50 841, EC50 476, Kd 3
77	OXTR	P30559	1,306	1,182	31	0.359	354	0.714	7	Ki 701, EC50 338, IC50 232, Kd 35
78	TBXA2R	P21731	1,305	1,257	5	0.333	3	0.500	10	IC50 577, Ki 456, Kd 227, EC50 45
79	CXCR2	P25025	1,295	1,260	92	0.655	2,344	0.796	49	IC50 1061, Ki 219, Kd 14, EC50 1
80	EDNRB	P24530	1,294	1,266	4	1.000	1	1.000	1	IC50 1097, Ki 187, Kd 5, Kb 4, EC50 1
81	CALCRL	Q16602	1,268	897	6	1.000	6	—	—	Ki 631, IC50 612, EC50 14, Kd 8, Kb 3
82	SSTR3	P32745	1,258	1,079	8	0.833	6	0.400	15	IC50 589, Ki 397, EC50 193, Kd 79
83	MTNR1B	P49286	1,247	1,029	66	0.664	1,452	0.873	63	Ki 925, EC50 182, IC50 97, Kb 40, Kd 3
84	GRM1	Q13255	1,242	1,132	27	0.770	270	0.667	12	IC50 866, EC50 263, Ki 97, Kb 16
85	PTGER3	P43115	1,230	1,068	7	1.000	4	1.000	8	IC50 553, Ki 536, EC50 131, Kb 10
86	SSTR5	P35346	1,220	1,172	35	0.617	350	0.385	13	IC50 717, Ki 396, EC50 73, Kd 34
87	GPBAR1	Q8TDU6	1,189	1,182	171	0.763	4,867	—	—	EC50 1155, IC50 34
88	CCR3	P51677	1,187	1,177	10	0.422	45	—	—	IC50 769, Ki 408, EC50 5, Kb 3, Kd 2
89	C5AR1	P21730	1,166	1,074	151	0.673	5,017	0.406	64	IC50 1061, EC50 55, Ki 50
90	PTGER1	P34995	1,160	1,020	6	—	—	1.000	8	IC50 674, Ki 414, EC50 48, Kd 14, Kb 10
91	ADRA2A	P08913	1,158	1,027	216	0.682	7,619	0.643	1,033	Ki 809, IC50 148, EC50 127, Kb 69, Kd 5
92	PTGER2	P43116	1,154	1,032	50	0.495	858	0.958	48	Ki 422, EC50 356, Kb 196, IC50 176, Kd 4
93	TACR2	P21452	1,147	1,118	1	—	—	1.000	5	Ki 853, IC50 277, Kd 11, EC50 5, Kb 1
94	BDKRB1	P46663	1,147	890	4	1.000	2	1.000	1	Ki 702, IC50 441, Kd 2, Kb 2
95	NPY1R	P25929	1,132	999	18	0.667	6	0.857	28	Ki 658, IC50 350, Kb 63, EC50 40, Kd 21
96	AVPR2	P30518	1,124	1,049	85	0.416	2,650	0.808	52	Ki 454, IC50 374, EC50 286, Kd 10
97	AGTR1	P30556	1,087	1,044	71	0.500	969	0.670	109	IC50 751, Ki 199, EC50 103, Kd 25, Kb 9
98	F2R	P25116	1,053	992	23	0.818	22	0.952	21	IC50 848, EC50 112, Ki 78, Kd 15
99	P2RY1	P47900	1,024	884	11	0.684	19	0.692	13	Ki 711, IC50 237, EC50 68, Kd 6, Kb 2
100	HTR4	Q13639	991	793	63	0.653	1,073	—	—	Ki 496, EC50 389, IC50 91, Kb 12, Kd 3
101	CCR1	P32246	985	936	3	1.000	1	1.000	1	IC50 803, Ki 160, EC50 21, Kd 1
102	HCAR2	Q8TDS4	955	737	1	—	—	1.000	1	EC50 631, IC50 291, Ki 33
103	GPR6	P46095	946	941	3	—	—	0.000	3	IC50 546, EC50 396, Ki 4
104	ADRA2C	P18825	926	743	95	0.659	2,950	0.632	775	Ki 629, EC50 152, IC50 73, Kb 72
105	PTGDR	Q13258	908	819	0	—	—	—	—	IC50 449, Ki 329, EC50 65, Kb 64, Kd 1
106	NPY2R	P49146	905	776	23	0.818	22	0.875	32	IC50 414, Ki 288, EC50 187, Kd 15, Kb 1
107	HRH2	P25021	883	751	25	0.602	171	0.559	177	Ki 559, EC50 148, IC50 91, Kd 66, Kb 19
108	SSTR1	P30872	878	867	19	0.661	56	0.682	22	IC50 547, Ki 261, Kd 58, EC50 12
109	AVPR1B	P47901	868	857	9	0.952	21	1.000	6	IC50 412, Ki 246, EC50 204, Kd 6
110	SMO	Q99835	857	831	6	0.667	6	—	—	IC50 812, EC50 22, Ki 17, Kd 6
111	FFAR2	O15552	852	828	25	0.611	275	—	—	EC50 651, IC50 173, Ki 28
112	AGTR2	P50052	814	802	41	0.638	639	0.929	14	IC50 604, Ki 210
113	FPR1	P21462	793	733	112	0.583	3,031	0.502	221	EC50 552, IC50 184, Kd 43, Ki 14
114	UTS2R	Q9UKP6	768	687	2	1.000	1	—	—	Ki 324, EC50 240, IC50 198, Kd 6
115	CCKAR	P32238	749	517	3	—	—	—	—	IC50 347, EC50 206, Ki 195, Kd 1
116	S1PR2	O95136	738	719	4	0.500	2	1.000	7	IC50 570, EC50 92, Kd 75, Ki 1
117	CCR4	P51679	731	658	0	—	—	—	—	IC50 578, Ki 99, Kd 45, EC50 9
118	GPR84	Q9NQS5	716	683	315	0.569	9,942	—	—	IC50 505, EC50 135, Ki 73, Kb 2, Kd 1
119	PTGIR	P43119	697	646	0	—	—	—	—	Ki 280, IC50 189, EC50 179, Kb 49
120	BDKRB2	P30411	687	591	2	—	—	1.000	2	Ki 329, IC50 250, Kd 106, EC50 2
121	NTSR1	P30989	675	584	20	0.754	69	0.500	8	EC50 371, Ki 164, IC50 129, Kd 11
122	S1PR4	O95977	661	649	2	1.000	1	1.000	8	IC50 383, EC50 267, Kd 8, Ki 2, Kb 1
123	S1PR5	Q9H228	647	632	4	0.833	6	0.875	8	EC50 376, IC50 258, Kd 8, Ki 5
124	ADRA2B	P18089	641	539	128	0.631	3,610	0.592	817	Ki 488, EC50 76, IC50 40, Kb 37
125	CASR	P41180	628	628	31	0.426	434	—	—	IC50 396, EC50 232
126	PTGFR	P43088	628	617	0	—	—	—	—	IC50 466, Ki 97, EC50 65
127	DRD5	P21918	604	597	49	0.809	1,113	0.777	435	Ki 550, EC50 34, IC50 16, Kd 4
128	HTR5A	P47898	503	485	45	0.620	820	0.678	537	Ki 453, IC50 45, Kd 3, EC50 2
129	GPR35	Q9HC97	501	310	96	0.613	1,647	0.593	209	EC50 295, IC50 146, Ki 59, Kd 1
130	LPAR1	Q92633	487	432	240	0.611	5,583	0.209	67	IC50 340, Ki 56, EC50 51, Kb 36, Kd 4
131	FPR3	P25089	465	465	42	0.480	741	0.599	177	EC50 465
132	BRS3	P32247	457	340	36	0.611	267	0.667	9	EC50 319, IC50 136, Ki 2
133	LTB4R	Q15722	448	406	3	—	—	0.500	4	IC50 245, Ki 143, EC50 54, Kb 6
134	PTAFR	P25105	443	438	16	0.686	86	—	—	IC50 424, Ki 19
135	NPY4R	P50391	419	270	75	0.766	770	0.968	62	Ki 220, EC50 129, IC50 39, Kb 28, Kd 3
136	P2RY2	P41231	417	407	20	0.831	71	0.500	4	EC50 275, IC50 86, Kd 41, Ki 15
137	CXCR1	P25024	409	400	6	0.500	4	0.571	7	IC50 305, Ki 102, EC50 1, Kd 1
138	GPR139	Q6DWJ6	407	316	57	0.534	1,596	—	—	EC50 313, Ki 94
139	KISS1R	Q969F8	401	316	3	—	—	1.000	1	EC50 209, IC50 101, Ki 91
140	CCR9	P51686	398	396	2	0.000	1	—	—	IC50 263, Ki 134, EC50 1
141	CMKLR1	Q99788	370	339	83	0.510	1,629	0.750	4	IC50 320, EC50 50
142	P2RY6	Q15077	359	354	65	0.483	1,918	0.200	10	EC50 279, IC50 75, Ki 5
143	GRM3	Q14832	352	254	19	0.742	31	0.652	23	IC50 151, EC50 116, Ki 85
144	PRLHR	P49683	349	257	0	—	—	—	—	Ki 161, IC50 95, EC50 93
145	GPR88	Q9GZN0	336	336	63	0.567	1,601	—	—	EC50 336
146	TAS2R8	Q9NYW2	322	322	0	—	—	—	—	IC50 321, EC50 1
147	GPR52	Q9Y2T5	322	319	53	0.588	1,373	0.000	1	EC50 292, IC50 30
148	PROKR1	Q8TCW9	313	313	0	—	—	—	—	IC50 310, Ki 3
149	GPR55	Q9Y2T6	312	255	63	0.464	923	0.500	4	IC50 178, EC50 126, Kb 5, Kd 3
150	MRGPRX4	Q96LA9	309	309	0	—	—	—	—	IC50 309
151	P2RY14	Q15391	303	297	111	0.563	3,601	0.854	48	IC50 235, EC50 56, Ki 11, Kb 1
152	GRM7	Q14831	302	287	17	0.701	117	0.818	11	IC50 182, EC50 102, Ki 18
153	C3AR1	Q16581	278	218	12	—	—	0.500	20	IC50 169, EC50 108, Kd 1
154	TAAR1	Q96RJ0	277	243	87	0.502	3,252	0.111	9	EC50 224, Ki 50, IC50 3
155	CALCR	P30988	274	158	41	0.512	406	—	—	EC50 143, IC50 116, Ki 15
156	LPAR3	Q9UBY5	271	229	6	0.667	6	0.571	14	IC50 144, Ki 67, EC50 60
157	MLNR	O43193	268	245	1	—	—	1.000	1	EC50 149, Ki 93, IC50 26
158	CYSLTR1	Q9Y271	259	254	0	—	—	—	—	IC50 237, Kd 10, EC50 8, Ki 4
159	NPBWR1	P48145	249	239	0	—	—	—	—	IC50 200, EC50 48, Kb 1
160	P2RY4	P51582	242	240	4	0.800	5	0.500	4	EC50 164, IC50 77, Kb 1
161	F2RL1	P55085	241	238	4	0.000	2	—	—	EC50 126, IC50 112, Ki 3
162	HTR1E	P28566	240	240	16	0.448	105	0.748	218	Ki 228, IC50 12
163	GRPR	P30550	238	230	21	0.445	200	0.571	7	IC50 185, Ki 44, EC50 8, Kb 1
164	CCR8	P51685	223	213	50	0.282	1,067	—	—	IC50 130, Ki 75, EC50 18
165	GPR142	Q7Z601	221	221	0	—	—	—	—	EC50 174, IC50 47
166	NTSR2	O95665	209	197	9	0.750	28	0.500	8	Ki 122, EC50 53, IC50 32, Kd 2
167	HCAR1	Q9BXC0	198	198	6	0.667	15	1.000	1	EC50 198
168	GRM8	O00222	192	180	9	0.611	18	0.647	17	EC50 126, IC50 44, Ki 21, Kd 1
169	GPR18	Q14330	192	141	81	0.466	2,549	0.800	5	IC50 136, EC50 54, Kd 1, Kb 1
170	NMBR	P28336	185	177	1	—	—	—	—	Ki 104, IC50 71, EC50 8, Kb 2
171	GIPR	P48546	182	181	38	0.540	507	0.538	39	IC50 150, EC50 28, Ki 4
172	HTR1F	P30939	181	152	0	—	—	—	—	Ki 140, EC50 25, IC50 16
173	ADCYAP1R1	P41586	180	106	0	—	—	—	—	IC50 89, EC50 71, Ki 16, Kd 4
174	QRFPR	Q96P65	177	142	0	—	—	—	—	EC50 92, IC50 79, Ki 6
175	NPFFR2	Q9Y5X5	177	158	46	0.742	565	0.571	70	Ki 104, EC50 63, IC50 8, Kd 2
176	NMUR2	Q9GZQ4	176	130	4	1.000	2	1.000	4	EC50 125, IC50 47, Ki 4
177	CCR6	P51684	175	174	67	0.755	1,844	0.500	4	IC50 174, EC50 1
178	LPAR5	Q9H1C0	172	170	3	1.000	1	0.286	7	IC50 158, EC50 13, Ki 1
179	GRM6	O15303	170	159	3	1.000	1	0.625	8	EC50 109, IC50 36, Ki 25
180	LPAR2	Q9HBW0	169	163	62	0.282	1,813	0.162	68	IC50 100, EC50 61, Ki 7, Kd 1
181	NPFFR1	Q9GZQ6	168	148	38	0.690	538	0.792	48	Ki 99, EC50 54, IC50 8, Kd 5, Kb 2
182	PTH1R	Q03431	167	150	0	—	—	—	—	EC50 76, IC50 59, Ki 26, Kd 6
183	MCHR2	Q969V1	158	157	0	—	—	—	—	Ki 94, IC50 64
184	MRGPRX1	Q96LB2	157	157	1	—	—	—	—	EC50 125, IC50 32
185	CCRL2	O00421	154	154	0	—	—	—	—	IC50 154
186	NMUR1	Q9HB89	141	98	4	1.000	2	1.000	4	EC50 90, IC50 47, Ki 4
187	GPR183	P32249	130	130	143	0.479	4,685	0.485	233	IC50 124, EC50 6
188	HCAR3	P49019	127	126	0	—	—	—	—	EC50 123, IC50 4
189	RXFP3	Q9NSD7	127	104	33	0.535	256	0.210	19	EC50 68, Ki 32, IC50 27
190	GPR34	Q9UPC5	123	123	25	0.689	180	—	—	IC50 79, EC50 44
191	GPR17	Q13304	122	118	96	0.568	3,163	—	—	EC50 69, IC50 46, Ki 6, Kd 1
192	TAS2R14	Q9NYV8	121	120	33	0.562	525	—	—	IC50 117, EC50 4
193	GPER1	Q99527	120	116	2	—	—	—	—	IC50 111, EC50 5, Ki 4
194	GLP2R	O95838	111	111	10	0.571	42	0.000	1	EC50 102, IC50 9
195	GALR1	P47211	110	106	0	—	—	—	—	IC50 63, Ki 40, Kd 7
196	RXFP1	Q9HBX9	110	108	144	0.594	4,963	0.778	9	EC50 105, Ki 5
197	CYSLTR2	Q9NS75	106	106	0	—	—	—	—	IC50 103, EC50 3
198	GPR174	Q9BXC1	104	98	0	—	—	—	—	EC50 97, IC50 7
199	FSHR	P23945	95	95	30	0.581	425	1.000	29	EC50 64, IC50 31
200	VIPR2	P41587	89	87	0	—	—	—	—	EC50 53, IC50 36
201	NPSR1	Q6W5P4	88	87	0	—	—	—	—	IC50 86, EC50 1, Ki 1
202	GPR39	O43194	87	85	0	—	—	—	—	EC50 87
203	FFAR3	O14843	86	85	6	0.333	15	—	—	EC50 85, IC50 1
204	GALR2	O43603	84	81	0	—	—	—	—	IC50 39, Ki 38, Kd 7
205	CRHR2	Q13324	79	73	0	—	—	—	—	IC50 63, Ki 10, EC50 6
206	OXER1	Q8TDS5	78	77	0	—	—	—	—	IC50 71, EC50 7
207	CXCR5	P32302	77	76	1	—	—	—	—	IC50 76, EC50 1
208	GPR4	P46093	75	75	0	—	—	—	—	IC50 75
209	MRGPRX2	Q96LB1	71	71	8	0.000	1	—	—	EC50 65, IC50 6
210	LHCGR	P22888	69	67	9	0.500	12	0.429	7	IC50 37, EC50 31, Ki 1
211	RXFP4	Q8TDU9	67	45	24	0.547	95	0.167	18	EC50 42, Ki 22, IC50 3
212	CX3CR1	P49238	66	65	32	0.462	238	0.625	120	Ki 51, IC50 14, EC50 1
213	SUCNR1	Q9BXA5	66	66	48	0.484	355	—	—	IC50 66
214	CXCR6	O00574	64	63	0	—	—	—	—	IC50 63, EC50 1
215	LTB4R2	Q9NPC1	60	59	56	0.563	584	0.625	8	EC50 53, IC50 6, Kd 1
216	GPR65	Q8IYL9	57	57	41	0.503	752	0.532	203	IC50 55, EC50 2
217	P2RY10	O00398	51	51	14	0.736	91	—	—	EC50 51
218	CCR10	P46092	51	51	0	—	—	—	—	IC50 51
219	TSHR	P16473	49	49	38	0.514	440	0.938	32	IC50 29, EC50 20
220	VIPR1	P32241	49	46	0	—	—	—	—	EC50 36, IC50 12, Ki 1
221	P2RY11	Q96G91	49	46	0	—	—	—	—	EC50 31, Ki 15, IC50 3
222	FZD7	O75084	40	35	1	—	—	—	—	Kd 35, IC50 5
223	TRHR	P34981	36	18	0	—	—	—	—	Ki 18, EC50 18
224	GPR27	Q9NS67	32	32	30	0.505	414	—	—	EC50 32
225	GALR3	O60755	30	30	0	—	—	—	—	Ki 26, Kd 4
226	OR51E2	Q9H255	24	24	0	—	—	—	—	EC50 23, IC50 1
227	LPAR4	Q99677	17	17	4	0.333	3	0.182	11	EC50 13, Ki 2, IC50 2
228	TAS2R46	P59540	16	15	0	—	—	—	—	EC50 10, IC50 6
229	P2RY13	Q9BPV8	15	15	0	—	—	—	—	EC50 9, IC50 6
230	TAS2R31	P59538	14	14	0	—	—	—	—	EC50 8, IC50 6
231	CCR7	P32248	12	11	72	0.509	1,140	0.800	40	IC50 11, EC50 1
232	TAS2R38	P59533	12	12	0	—	—	—	—	EC50 12
233	GPR68	Q15743	12	12	1	—	—	—	—	EC50 10, IC50 2
234	LPAR6	P43657	11	11	0	—	—	—	—	EC50 11
235	SCTR	P47872	11	10	2	1.000	1	1.000	2	EC50 10, Ki 1
236	TAS2R16	Q9NYV7	11	10	0	—	—	—	—	EC50 10, IC50 1
237	PROKR2	Q8NFJ6	8	8	0	—	—	—	—	Ki 8
238	OXGR1	Q96P68	8	8	0	—	—	—	—	IC50 8
239	GABBR1	Q9UBS5	8	7	0	—	—	—	—	EC50 6, Ki 1, IC50 1
240	TAS2R10	Q9NYW0	6	6	0	—	—	—	—	EC50 6
241	FZD1	Q9UP38	5	5	0	—	—	—	—	Kd 3, IC50 1, EC50 1
242	CMKLR2	P46091	4	4	5	0.750	4	0.750	4	EC50 4
243	C5AR2	Q9P296	4	2	14	—	—	0.375	24	Ki 2, EC50 2
244	TAS2R60	P59551	3	3	0	—	—	—	—	EC50 3
245	TAS2R9	Q9NYW1	3	3	0	—	—	—	—	EC50 3
246	TAS2R4	Q9NYW5	3	3	0	—	—	—	—	EC50 3
247	TAS2R1	Q9NYW7	3	3	0	—	—	—	—	EC50 3
248	ACKR2	O00590	2	1	5	—	—	1.000	5	EC50 1, IC50 1
249	MAS1	P04201	2	2	0	—	—	—	—	IC50 2
250	TAS2R41	P59536	2	2	0	—	—	—	—	EC50 2
251	TAS2R43	P59537	2	2	0	—	—	—	—	EC50 2
252	FZD2	Q14332	2	2	0	—	—	—	—	IC50 1, EC50 1
253	TAS2R13	Q9NYV9	2	2	0	—	—	—	—	EC50 2
254	TAAR5	O14804	1	1	0	—	—	—	—	EC50 1
255	GPR37L1	O60883	1	1	0	—	—	—	—	IC50 1
256	ADGRE5	P48960	1	1	0	—	—	—	—	Kd 1
257	GPR15	P49685	1	1	0	—	—	—	—	EC50 1
258	TAS2R39	P59534	1	1	0	—	—	—	—	EC50 1
259	TAS2R40	P59535	1	1	0	—	—	—	—	EC50 1
260	TAS2R45	P59539	1	1	0	—	—	—	—	EC50 1
261	TAS2R30	P59541	1	1	0	—	—	—	—	EC50 1
262	TAS2R19	P59542	1	1	0	—	—	—	—	EC50 1
263	TAS2R20	P59543	1	1	0	—	—	—	—	EC50 1
264	TAS2R50	P59544	1	1	0	—	—	—	—	EC50 1
265	MC2R	Q01718	1	1	37	0.682	340	—	—	IC50 1
266	GHRHR	Q02643	1	1	0	—	—	—	—	IC50 1
267	OR10J3	Q5JRS4	1	1	0	—	—	—	—	Kd 1
268	TAS2R42	Q7RTR8	1	1	0	—	—	—	—	EC50 1
269	GPR135	Q8IZ08	1	1	0	—	—	—	—	EC50 1
270	TAS2R7	Q9NYW3	1	1	0	—	—	—	—	EC50 1
271	TAS2R5	Q9NYW4	1	1	0	—	—	—	—	EC50 1
272	TAS2R3	Q9NYW6	1	1	0	—	—	—	—	EC50 1
273	GPR3	P46089	0	0	53	0.605	1,079	0.000	3
274	GPR143	P51810	0	0	1	—	—	—	—
275	ADGRF1	Q5T601	0	0	26	0.700	130	0.530	132
276	MRGPRX3	Q96LB0	0	0	1	—	—	—	—
277	LGR4	Q9BXB1	0	0	1	—	—	0.000	2
278	GPR132	Q9UNW8	0	0	36	0.619	627	1.000	2